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辛波莫德半富馬酸鹽

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Siponimod Hemifumarate (Synonyms: BAF-312 Hemifumarate)

產(chǎn)品編號(hào):CL1367A CAS No.:1234627-85-0 MDLNo: 分子式:C29H35F3N2O3·1/2C4H4O4 分子量:574.63 | 516.61(free)
規(guī)格 庫(kù)存 目錄價(jià) 會(huì)員專享價(jià) 數(shù)量
5 mg 3-5days ¥1166.00 登錄后可見(jiàn)
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10 mg 3-5days ¥1800.00 登錄后可見(jiàn)
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基本信息
英文名稱 Siponimod Hemifumarate (Synonyms: BAF-312 Hemifumarate)
中文名稱辛波莫德半富馬酸鹽
CAS號(hào)1234627-85-0
分子式C29H35F3N2O3·1/2C4H4O4
分子量574.63 | 516.61(free)
產(chǎn)品詳情

Siponimod (BAF-312) hemifumarate is a potent and selective sphingosine-1-phosphate (S1P) receptor modulator. Siponimod hemifumarate is selective for S1P1 and S1P5 receptors over S1P2, S1P3, and S1P4 (EC50s of 0.39, 0.98, >10000, >1000, and 750 nM, respectively). Siponimod hemifumarate can be used for multiple sclerosis (MS) research.
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相關(guān)文獻(xiàn)

Prospects of siponimod in secondary progressive multiple sclerosis.

PMID: 30038666 PMCID: PMC6050809 DOI: 10.1177/1756286418788013

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