英文名稱 | Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride) |
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中文名稱 | Olcegepant hydrochloride (BIBN-4096 hydrochloride; BIBN4096BS hydrochloride) |
CAS號 | 586368-06-1 |
分子式 | C38H47Br2N9O5.HCl |
分子量 | 906.11 |
英文名稱 | Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride) |
---|---|
中文名稱 | Olcegepant hydrochloride (BIBN-4096 hydrochloride; BIBN4096BS hydrochloride) |
CAS號 | 586368-06-1 |
分子式 | C38H47Br2N9O5.HCl |
分子量 | 906.11 |
Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.