英文名稱 | MYCi975 (Synonyms:NUCC-0200975) |
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中文名稱 | MYCi975 (NUCC-0200975) |
CAS號 | 2289691-01-4 |
分子式 | C25H16Cl2F6N2O2 |
分子量 | 561.30 |
英文名稱 | MYCi975 (Synonyms:NUCC-0200975) |
---|---|
中文名稱 | MYCi975 (NUCC-0200975) |
CAS號 | 2289691-01-4 |
分子式 | C25H16Cl2F6N2O2 |
分子量 | 561.30 |
MYCi975 (NUCC-0200975) is a potent, selective and orally active inhibitor of MYC that disrupts MYC/MAX interaction, promotes MYC T58 phosphorylation and MYC degradation, and impairs MYC driven gene expression. MYCi975 exhibits potent anti-tumor activities.
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